The Experts below are selected from a list of 1014 Experts worldwide ranked by ideXlab platform
Jean M. Schmidt - One of the best experts on this subject based on the ideXlab platform.
-
Antineoplastic agents. 520. Isolation and structure of Irciniastatins A and B from the Indo-Pacific marine sponge Ircinia ramosa.
Journal of medicinal chemistry, 2004Co-Authors: George R. Pettit, Jean-charles Chapuis, Robin K. Pettit, Larry P. Tackett, Dennis L. Doubek, John N. A. Hooper, Jean M. SchmidtAbstract:The Indo-Pacific marine sponge Ircinia ramosa has been found to contain two powerful (GI50 from 0.001 to
-
antineoplastic agents 520 isolation and structure of Irciniastatins a and b from the indo pacific marine sponge Ircinia ramosa
Journal of Medicinal Chemistry, 2004Co-Authors: George R. Pettit, Jean-charles Chapuis, Robin K. Pettit, Larry P. Tackett, Dennis L. Doubek, John N. A. Hooper, Jean M. SchmidtAbstract:The Indo-Pacific marine sponge Ircinia ramosa has been found to contain two powerful (GI50 from 0.001 to <0.0001 μg/mL) murine and human cancer cell growth inhibitors. Both were isolated (10-3−10-4% yields) by cancer cell line bioassay-guided techniques and named Irciniastatins A (1) and B (2). Structural elucidation by a combination of spectral analyses, primarily high resolution mass and 2D-NMR (principally APT, HMQC, HMBC, and ROESY) spectroscopy, revealed the unusual structures 1 and 2.
Guido Cimino - One of the best experts on this subject based on the ideXlab platform.
-
wistarin from the marine sponge Ircinia sp the first case of enantiomeric sesterterpenes
Tetrahedron-asymmetry, 1999Co-Authors: Angelo Fontana, Issa M. I. Fakhr, Ernesto Mollo, Guido CiminoAbstract:Abstract The sestertepene (−)-wistarin has been isolated from a Red Sea sponge of the genus Ircinia . This metabolite is the enantiomer of (+)-wistarin, a tetracyclic metabolite previously isolated from the sponge Ircinia wistarii . The enantiomeric relationship was proved by comparison of the CD spectrum of (−)-wistarin with that of a synthetic sample of the (+)-isomer. A hypothetical biosynthesis of (−)-wistarin is discussed starting from a putative linear precursor.
-
(−)-Wistarin from the marine sponge Ircinia sp.: the first case of enantiomeric sesterterpenes
Tetrahedron: Asymmetry, 1999Co-Authors: Angelo Fontana, Issa M. I. Fakhr, Ernesto Mollo, Guido CiminoAbstract:Abstract The sestertepene (−)-wistarin has been isolated from a Red Sea sponge of the genus Ircinia . This metabolite is the enantiomer of (+)-wistarin, a tetracyclic metabolite previously isolated from the sponge Ircinia wistarii . The enantiomeric relationship was proved by comparison of the CD spectrum of (−)-wistarin with that of a synthetic sample of the (+)-isomer. A hypothetical biosynthesis of (−)-wistarin is discussed starting from a putative linear precursor.
Pei-show Shih - One of the best experts on this subject based on the ideXlab platform.
-
irciformonins e k c22 trinorsesterterpenoids from the sponge Ircinia formosana
Helvetica Chimica Acta, 2009Co-Authors: Ya-ching Shen, Yu-chi Lin, Yao-haur Kuo, Pei-show Shih, Yun-sheng Lin, Yuh-chi Kuo, Ashraf Taha KhalilAbstract:Chemical investigation of the sponge Ircinia formosana resulted in the isolation of seven new linear C22-sesterterpenoids, irciformonins E–K (1–7) in addition to irciformonin A (8), a previously isolated furanosesterterpenoid (=a furan-moiety-containing sesterterpenoid) from the same species. The structures were determined by interpretation of HR-ESI-MS and 2D-NMR spectra. The structure of irciformonin A (8) was revised. Compound 5 exhibited significant inhibition of peripheral blood mononuclear cell proliferation induced by phytohemaglutinin.
-
Irciformonins E – K, C22‐Trinorsesterterpenoids from the Sponge Ircinia formosana
Helvetica Chimica Acta, 2009Co-Authors: Ya-ching Shen, Yu-chi Lin, Yao-haur Kuo, Pei-show Shih, Yun-sheng Lin, Yuh-chi Kuo, Ashraf Taha KhalilAbstract:Chemical investigation of the sponge Ircinia formosana resulted in the isolation of seven new linear C22-sesterterpenoids, irciformonins E–K (1–7) in addition to irciformonin A (8), a previously isolated furanosesterterpenoid (=a furan-moiety-containing sesterterpenoid) from the same species. The structures were determined by interpretation of HR-ESI-MS and 2D-NMR spectra. The structure of irciformonin A (8) was revised. Compound 5 exhibited significant inhibition of peripheral blood mononuclear cell proliferation induced by phytohemaglutinin.
-
Novel linear C22-sesterterpenoids from sponge Ircinia formosana
Tetrahedron Letters, 2006Co-Authors: Ya-ching Shen, Yu-chi Lin, Ashraf Taha Khalil, Yao-haur Kuo, Pei-show ShihAbstract:Abstract Four unprecedented C 22 -sesterterpenes, irciformonins A–D ( 1 – 4 ), have been isolated from the marine sponge Ircinia formosana , collected off the coast of eastern Taiwan. The structures of the isolated metabolites were established on the basis of extensive spectral analysis, primarily 1- and 2D-NMR. Compounds 3 and 4 exhibited significant cytotoxicity against human colon (WiDr) tumor cells.
S. De Rosa - One of the best experts on this subject based on the ideXlab platform.
-
Lipophylic metabolites from the marine sponge Ircinia muscarum and its cell cultures
Marine Biology, 2002Co-Authors: S. De Rosa, Giuseppina Tommonaro, Krasimir Slantchev, Kamen Stefanov, Simeon PopovAbstract:The composition of the lipophylic extract from the sponge Ircinia muscarum and its cell cultures developed under light and dark conditions was investigated. Lipids and their fatty acids, as well as volatile compounds and sterols, were identified. The differences between the two cell cultures did not appear to be very significant, while there were significant differences between the sponge and the cell cultures. Most of the isolated compounds were found for the first time in dictyoceratide sponges.
-
Palinurin and Fasciculatin Sulfates from Two Thyrrenean Sponges of the Genus Ircinia
Natural Product Letters, 1997Co-Authors: S. De Rosa, A. De Giulio, A. Crispino, Carmine Iodice, Giuseppina TommonaroAbstract:Abstract Together with the previously described palinurin (1a) and fasciculatin (2a), the corresponding sulfates 1b and 2b were isolated from sponges of the genus Ircinia, collected in the Thyrrenean Sea. The structural elucidation and biological activity of these compounds are reported.
-
Sulfated Furanosesterterpenes from Two Sponges of the Genus Ircinia
Natural Product Letters, 1996Co-Authors: S. De Rosa, A. Milone, A. De Giulio, A. Crispino, Carmine IodiceAbstract:Abstract Together with the previously described (18R)-variabilin (1a), its 13Z-isomer 2a, ircinin 1 (3a) and ircinin 2 (4a), the corresponding sulfates 1b-4b were isolated from sponges of the genus Ircinia, collected in the Northern Adriatic Sea. The structural elucidation and biological activity of these compounds are reported.
-
Pharmacological studies on terpenoids from marine sponges: Analgesic and muscle relaxant effects
Phytotherapy Research, 1991Co-Authors: R. De Pasquale, S. De Rosa, C. Circosta, Francesco Occhiuto, S. De StefanoAbstract:Some terpenoids extracted from marine sponge: triacetylated desidein (from Disidea pallescens), 2-tetraprenyl benzoquinol and 4-hydroxy-3-tetraprenylbenzoic acid (from Ircinia muscarum), 2-polyprenyl benzoquinols (from Ircinia spinosula), avarol (from Disidea avara) and furospongin-1 (from Spongia officinalis) were tested by multidimensional Irwin screening and with some tests for analgesic and muscle relaxant activity. The three prenylhydroquinols derivatives and avarol show a good analgesic activity and low toxicity.
George R. Pettit - One of the best experts on this subject based on the ideXlab platform.
-
Antineoplastic agents. 520. Isolation and structure of Irciniastatins A and B from the Indo-Pacific marine sponge Ircinia ramosa.
Journal of medicinal chemistry, 2004Co-Authors: George R. Pettit, Jean-charles Chapuis, Robin K. Pettit, Larry P. Tackett, Dennis L. Doubek, John N. A. Hooper, Jean M. SchmidtAbstract:The Indo-Pacific marine sponge Ircinia ramosa has been found to contain two powerful (GI50 from 0.001 to
-
antineoplastic agents 520 isolation and structure of Irciniastatins a and b from the indo pacific marine sponge Ircinia ramosa
Journal of Medicinal Chemistry, 2004Co-Authors: George R. Pettit, Jean-charles Chapuis, Robin K. Pettit, Larry P. Tackett, Dennis L. Doubek, John N. A. Hooper, Jean M. SchmidtAbstract:The Indo-Pacific marine sponge Ircinia ramosa has been found to contain two powerful (GI50 from 0.001 to <0.0001 μg/mL) murine and human cancer cell growth inhibitors. Both were isolated (10-3−10-4% yields) by cancer cell line bioassay-guided techniques and named Irciniastatins A (1) and B (2). Structural elucidation by a combination of spectral analyses, primarily high resolution mass and 2D-NMR (principally APT, HMQC, HMBC, and ROESY) spectroscopy, revealed the unusual structures 1 and 2.